SCHEMBL5866623

SCHEMBL5866623

COC(=O)CC1(CS(=O)(=O)c2ccc(OCc3cc(C)nc4ccccc34)cc2)CCCC1

nearest known ligand 0.84

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 16/20 0.84
MMP13 P45452 9/20 0.84
MMP2 P08253 4/20 0.84
MMP9 P14780 2/20 0.84

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6794928 0.91 ADAM17 (1.00) ADAM17MMP13MMP2MMP9
SCHEMBL6795271 0.91 ADAM17 (1.00) ADAM17MMP13MMP2MMP9
SCHEMBL6788849 0.90 ADAM17 (1.00) ADAM17MMP13MMP2MMP9
Trifluoroacetic Acid SCHEMBL6787337 0.87 ADAM17 (0.91) ADAM17MMP13MMP2MMP9
Trifluoroacetic Acid SCHEMBL6794294 0.86 ADAM17 (0.91) ADAM17MMP13MMP2MMP9
SCHEMBL6787341 0.85 ADAM17 (0.77) ADAM17MMP13MMP2MMP9
Trifluoroacetic Acid SCHEMBL6790603 0.85 ADAM17 (0.91) ADAM17MMP13MMP2MMP9
SCHEMBL6794297 0.85 ADAM17 (0.78) ADAM17MMP13MMP2MMP9
SCHEMBL6790608 0.84 ADAM17 (0.77) ADAM17MMP13MMP2MMP9
SCHEMBL6794665 0.84 ADAM17 (1.00) ADAM17MMP13MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7074810-B2 Triazolone and triazolethione derivatives as inhibitors of matrix metalloproteinases and/or TNF-α converting enzyme BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-11 US disclosed
US-20040116491-A1 Triazolone and triazolethione derivatives as inhibitors of matrix metalloproteinases and/or TNF-alpha converting enzyme BRISTOL-MYERS SQUIBB COMPANY 2004-06-17 US disclosed