SCHEMBL5872364

SCHEMBL5872364

CC(C)C[C@H](N)C(F)(c1ccccc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
TAAR1 Q96RJ0 3/20 0.36
SLC6A2 P23975 2/20 0.36
MAOA P21397 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
CYP2A6 P11509 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
ANPEP P15144 1/20 0.36
LAP3 P28838 1/20 0.36
TACR1 P25103 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16635566 1.00 HTR2A (0.40) HTR2AHTR2CHTR2BALDH1A1TSHR
SCHEMBL635649 0.78 CYP2D6 (0.40) KDM4ELMNAMAPK1TAAR1SLC6A2
SCHEMBL1167957 0.77 ALDH1A1 (0.46) HTR2AHTR2CHTR2BALDH1A1TSHR
SCHEMBL1131722 0.77 KDM4E (0.58) ALDH1A1KDM4ELMNAMAPK1TAAR1
SCHEMBL4918492 0.77 KDM4E (0.58) ALDH1A1KDM4ELMNAMAPK1TAAR1
SCHEMBL1131718 0.77 KDM4E (0.58) ALDH1A1KDM4ELMNAMAPK1TAAR1
Hydrochloric Acid SCHEMBL8841082 0.76 KDM4E (0.56) ALDH1A1KDM4ELMNAMAPK1ANPEP
Hydrochloric Acid SCHEMBL8841083 0.76 KDM4E (0.56) ALDH1A1KDM4ELMNAMAPK1ANPEP
SCHEMBL7158095 0.74 CYP2D6 (0.37) KDM4ELMNAMAPK1TAAR1SLC6A2
SCHEMBL4521336 0.73 CYP2D6 (0.53) KDM4ELMNAMAPK1TAAR1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1135349-B1 PROCESS FOR PREPARING CHIRAL COMPOUNDS UNIV ST ANDREWS (GB) 2005-04-06 EP claimed
US-7126028-B1 Process for preparing chiral compounds THE UNIVERSITY COURT OF THE UNIVERSITY OF ST. ANDREWS (GB) 2006-10-24 US disclosed
EP-1135349-B1 PROCESS FOR PREPARING CHIRAL COMPOUNDS UNIV ST ANDREWS (GB) 2005-04-06 EP disclosed
EP-1135349-A1 PROCESS FOR PREPARING CHIRAL COMPOUNDS UNIVERSITY OF DURHAM (GB) 2001-09-26 EP disclosed
WO-2000034210-A1 PROCESS FOR PREPARING CHIRAL COMPOUNDS UNIVERSITY OF DURHAM (GB) 2000-06-15 WO disclosed