SCHEMBL587423

SCHEMBL587423

COC(=O)C1CCN(C(=O)OC)C(Cc2cccc(C(F)(F)F)c2)C1.COC(=O)N1CCC(C(=O)O)CC1Cc1cccc(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 6/20 0.45
NOTUM Q6P988 1/20 0.43
S1PR1 P21453 3/20 0.42
S1PR5 Q9H228 3/20 0.42
GRK5 P34947 1/20 0.42
CDK8 P49336 1/20 0.42
PDGFRA P16234 2/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SIGMAR1 Q99720 2/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HRH3 Q9Y5N1 1/20 0.40
PIM1 P11309 1/20 0.40
CETP P11597 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581110 0.96 TACR1 (0.48) TACR1NOTUMS1PR1S1PR5GRK5
SCHEMBL586714 0.96 TACR1 (0.46) TACR1TSHRKMT2AALDH1A1SMN1; SMN2
SCHEMBL587559 0.88 TACR1 (0.43) TACR1NOTUMKMT2AALDH1A1MAPT
SCHEMBL580937 0.86 TACR1 (0.41) TACR1NOTUMS1PR1S1PR5GRK5
SCHEMBL3075266 0.85 TACR1 (0.50) TACR1NOTUMS1PR1S1PR5GRK5
SCHEMBL581282 0.84 TACR1 (0.46) TACR1NOTUMKMT2ASIGMAR1MAPT
SCHEMBL581527 0.84 TACR1 (0.46) TACR1NOTUMKMT2ASIGMAR1MAPT
SCHEMBL581783 0.84 TACR1 (0.46) TACR1NOTUMKMT2ASIGMAR1MAPT
SCHEMBL586823 0.84 TACR1 (0.44) TACR1KMT2AALDH1A1SMN1; SMN2MAPT
SCHEMBL581526 0.84 TACR1 (0.46) TACR1NOTUMKMT2ASIGMAR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed