SCHEMBL587559

SCHEMBL587559

COC(=O)C1CCN(C(=O)OC)C(Cc2ccc(C(F)(F)F)cc2)C1.COC(=O)N1CCC(C(=O)O)CC1Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.43
NOTUM Q6P988 1/20 0.41
CYP3A4 P08684 3/20 0.41
MAPT P10636 3/20 0.41
MAPK1 P28482 1/20 0.41
OPRK1 P41145 1/20 0.41
KDM4E B2RXH2 2/20 0.39
KMT2A Q03164 1/20 0.39
ATM Q13315 1/20 0.39
ALDH1A1 P00352 3/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581783 0.96 TACR1 (0.46) TACR1NOTUMCYP3A4MAPTMAPK1
SCHEMBL581282 0.96 TACR1 (0.46) TACR1NOTUMCYP3A4MAPTMAPK1
SCHEMBL581526 0.96 TACR1 (0.46) TACR1NOTUMCYP3A4MAPTMAPK1
SCHEMBL586823 0.96 TACR1 (0.44) TACR1CYP3A4MAPTMAPK1OPRK1
SCHEMBL581527 0.96 TACR1 (0.46) TACR1NOTUMCYP3A4MAPTMAPK1
SCHEMBL587423 0.88 TACR1 (0.45) TACR1NOTUMMAPTKMT2AALDH1A1
SCHEMBL581238 0.86 NPC1 (0.41) TACR1CYP3A4MAPK1KDM4EKMT2A
SCHEMBL588023 0.84 OPRK1 (0.45) CYP3A4MAPTOPRK1KMT2AALDH1A1
SCHEMBL580834 0.84 NOTUM (0.41) NOTUMCYP3A4MAPTKMT2AALDH1A1
SCHEMBL586614 0.84 ALDH1A1 (0.43) MAPTOPRK1KMT2AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed