SCHEMBL5875004

SCHEMBL5875004

O=c1nc2c(=O)n(Cc3ccccc3)c(=O)c-2n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 6/20 0.55
GSK3A P49840 1/20 0.55
GSK3B P49841 1/20 0.55
ALDH1A1 P00352 6/20 0.49
LMNA P02545 3/20 0.49
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
RECQL P46063 1/20 0.49
MAPK1 P28482 2/20 0.48
USP2 O75604 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48
HSD17B10 Q99714 1/20 0.48
POLB P06746 1/20 0.46
P2RX4 Q99571 1/20 0.46
KDM4E B2RXH2 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12895971 0.74 ALDH1A1 (0.58) CFTRGSK3AGSK3BALDH1A1LMNA
SCHEMBL8985073 0.74 GSK3B (0.67) GSK3AGSK3BALDH1A1LMNASMN1; SMN2
SCHEMBL22203802 0.74 SRC (0.62) GSK3AGSK3BALDH1A1LMNARAB9A
SCHEMBL14392803 0.74 ALDH1A1 (0.67) GSK3AGSK3BALDH1A1LMNARAB9A
SCHEMBL12895946 0.73 SRC (0.57) GSK3AGSK3BALDH1A1LMNARAB9A
SCHEMBL1729534 0.72 GSK3B (0.59) GSK3AGSK3BALDH1A1LMNASMN1; SMN2
SCHEMBL19032859 0.72 CFTR (1.00) CFTRALDH1A1LMNAMAPK1USP2
SCHEMBL29497996 0.72 CFTR (1.00) CFTRALDH1A1LMNAMAPK1USP2
SCHEMBL13259493 0.69 SRC (0.57) GSK3AGSK3BALDH1A1LMNARAB9A
SCHEMBL14472561 0.68 ALDH1A1 (0.50) GSK3AGSK3BALDH1A1LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006511564-A 2006-04-06 JP claimed
EP-1581477-A1 CYCLOALKENE DICARBOXYLIC ACID COMPOUNDS AS ANTI-INFLAMMATORY, IMMUNOMODULATORY AND ANTI-PROLIFERATORY AGENTS 4SC AG (DE) 2005-10-05 EP claimed
WO-2004056746-A1 CYCLOALKENE DICARBOXYLIC ACID COMPOUNDS AS ANTI-INFLAMMATORY, IMMUNOMODULATORY AND ANTI-PROLIFERATORY AGENTS 4SC AG (DE) 2004-07-08 WO claimed