SCHEMBL5877433

SCHEMBL5877433

COc1ccc(-c2nc3cc(Cl)ccc3c(=O)n2CC2CCCC(CN)C2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 4/20 0.46
EGFR P00533 1/20 0.45
POLB P06746 2/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
PDE4B Q07343 1/20 0.40
MAP3K11 Q16584 1/20 0.40
CYP2D6 P10635 3/20 0.39
HTR2C P28335 1/20 0.39
ALOX5 P09917 1/20 0.39
GHSR Q92847 2/20 0.39
CYP3A4 P08684 1/20 0.39
KCNH2 Q12809 1/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877641 0.93 ABCC1 (0.46) ABCC1POLBMEN1KMT2APDE4B
SCHEMBL5877840 0.91 EGFR (0.45) ABCC1EGFRPOLBMEN1KMT2A
SCHEMBL5877608 0.89 EGFR (0.48) ABCC1EGFRPOLBMEN1KMT2A
SCHEMBL5878318 0.88 ABCC1 (0.54) ABCC1POLBMEN1KMT2APDE4B
SCHEMBL5877717 0.88 EGFR (0.44) ABCC1EGFRPOLBMEN1KMT2A
SCHEMBL5877585 0.87 EGFR (0.52) ABCC1EGFRMEN1KMT2ACYP2D6
SCHEMBL5878215 0.87 EGFR (0.48) ABCC1EGFRPOLBMEN1KMT2A
SCHEMBL5878076 0.87 EGFR (0.46) ABCC1EGFRPOLBMEN1KMT2A
SCHEMBL5878313 0.86 PDE4B (0.43) ABCC1POLBMEN1KMT2APDE4B
SCHEMBL5877583 0.85 EGFR (0.53) ABCC1EGFRMEN1KMT2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed