SCHEMBL5878313

SCHEMBL5878313

COc1ccc(-c2nc3ccc(C)cc3c(=O)n2CC2CCCC(CN)C2)cc1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.43
ABCC1 P33527 2/20 0.42
POLB P06746 2/20 0.42
MAP3K11 Q16584 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
MAPK1 P28482 3/20 0.40
MAPT P10636 3/20 0.40
HSD17B10 Q99714 3/20 0.39
KDM4E B2RXH2 3/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
RAB9A P51151 1/20 0.39
CYP2D6 P10635 4/20 0.39
PDE10A Q9Y233 1/20 0.39
HTR2C P28335 1/20 0.39
HK1 P19367 1/20 0.39
HKDC1 Q2TB90 1/20 0.39
PNP P00491 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877568 0.92 F11 (0.46) PDE4BABCC1MAP3K11CYP2D6GHSR
SCHEMBL5877641 0.91 ABCC1 (0.46) PDE4BABCC1POLBMAP3K11MAPK1
SCHEMBL5877323 0.91 SMN1; SMN2 (0.45) PDE4BABCC1POLBMAP3K11KDM4E
SCHEMBL5878318 0.90 ABCC1 (0.54) PDE4BABCC1POLBALDH1A1HPGD
SCHEMBL5877963 0.89 ALDH1A1 (0.47) ABCC1POLBALDH1A1HPGDMAPK1
SCHEMBL5876953 0.89 ABCC1 (0.50) ABCC1ALDH1A1CYP2D6HTR2CMEN1
SCHEMBL5876985 0.87 CRHR1 (0.44) ABCC1POLBALDH1A1HPGDMAPK1
SCHEMBL5877811 0.87 ABCC1 (0.46) ABCC1TP53CYP2D6HTR2CKMT2A
SCHEMBL5877862 0.86 AVPR1B (0.46) ABCC1MAPTLMNA
SCHEMBL5877265 0.86 ABCC1 (0.44) ABCC1POLBALDH1A1HPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed