SCHEMBL5878463

SCHEMBL5878463

CC(C)(C)c1ccc(-c2nc3ccc(Cl)cc3c(=O)n2CC2CCCC(CN)C2)cc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.46
HTR2C P28335 1/20 0.46
GHSR Q92847 2/20 0.45
CYP3A4 P08684 1/20 0.45
KCNH2 Q12809 1/20 0.45
ALOX5 P09917 2/20 0.44
ABCC1 P33527 2/20 0.44
MAPT P10636 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
EGFR P00533 1/20 0.42
KDM4E B2RXH2 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
AVPR1A P37288 5/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877256 0.93 EGFR (0.48) CYP2D6HTR2CGHSRCYP3A4KCNH2
SCHEMBL5877579 0.91 ABCC1 (0.46) CYP2D6HTR2CGHSRCYP3A4KCNH2
SCHEMBL5877998 0.91 MEN1 (0.53) CYP2D6HTR2CGHSRCYP3A4KCNH2
SCHEMBL5878230 0.89 CYP2D6 (0.52) CYP2D6HTR2CGHSRCYP3A4KCNH2
SCHEMBL5878470 0.89 EGFR (0.53) CYP2D6HTR2CGHSRCYP3A4KCNH2
SCHEMBL5877009 0.88 F11 (0.47) CYP2D6GHSRKCNH2ABCC1MAPT
SCHEMBL5877561 0.87 CYP2D6 (0.46) CYP2D6HTR2CGHSRCYP3A4KCNH2
SCHEMBL5877973 0.85 CYP2D6 (0.47) CYP2D6HTR2CGHSRCYP3A4KCNH2
SCHEMBL5877392 0.85 CYP2D6 (0.46) CYP2D6HTR2CGHSRCYP3A4KCNH2
SCHEMBL5878159 0.85 AVPR1A (0.49) EGFRAVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed