Ethylenediamine

Ethylenediamine

SCHEMBL5884629

Cc1cnc(CNCCN)cn1.NCCN.NCCN.NCCN

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3PDE3APDE3BPDE4APDE4BPDE4CPDE4D

The experimentally established mechanism targets of Ethylenediamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 1/20 0.39
CYP1A2 P05177 16/20 0.37
CYP3A4 P08684 15/20 0.37
CLK4 Q9HAZ1 9/20 0.37
HSD17B10 Q99714 6/20 0.37
CYP2D6 P10635 4/20 0.37
CYP2C19 P33261 4/20 0.37
TSHR P16473 4/20 0.36
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
CYP2C9 P11712 1/20 0.35
MAPK1 P28482 1/20 0.35
ALDH1A1 P00352 5/20 0.35
TP53 P04637 1/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
CASP7 P55210 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5833062 0.98 CYP1A2 (0.38) TLR7CYP1A2CYP3A4CLK4HSD17B10
SCHEMBL5884618 0.95 TLR7 (0.36) TLR7CYP1A2CYP3A4CLK4HSD17B10
SCHEMBL24180048 0.80 CYP1A2 (0.42) CYP1A2CYP3A4CLK4HSD17B10CYP2D6
SCHEMBL5833413 0.80 CYP1A2 (0.38) CYP1A2CYP3A4CLK4HSD17B10CYP2D6
SCHEMBL25590589 0.79 HRH4 (0.42) TLR7CYP1A2CYP3A4CLK4HSD17B10
SCHEMBL2261177 0.77 CYP1A2 (0.40) CYP1A2CYP3A4CLK4HSD17B10CYP2D6
SCHEMBL7992424 0.76 SIRT6 (0.36) TLR7MEN1KMT2AALDH1A1TP53
SCHEMBL11365092 0.76 CYP3A4 (0.36) CYP1A2CYP3A4CLK4HSD17B10CYP2D6
SCHEMBL11365084 0.76 CYP3A4 (0.34) CYP1A2CYP3A4CLK4HSD17B10CYP2D6
SCHEMBL1196784 0.76 CYP1A2 (0.40) CYP1A2CYP3A4CLK4HSD17B10CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39140-E1 Heterocyclic compounds BAYER CROPSCIENCE K.K. (JP) 2006-06-20 US disclosed