SCHEMBL5884684

SCHEMBL5884684

NCCCN.NCCNCc1ccc(F)nc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MC4R P32245 2/20 0.42
MC5R P33032 2/20 0.42
MC3R P41968 1/20 0.41
CXCR4 P61073 1/20 0.40
CHRM2 P08172 2/20 0.40
HDAC1 Q13547 4/20 0.39
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
KAT2B Q92831 1/20 0.35
ROCK1 Q13464 1/20 0.35
SCN8A Q9UQD0 1/20 0.33
MAOB P27338 1/20 0.33
DYRK1A Q13627 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
NOS1 P29475 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5833046 0.97 MC4R (0.45) MC4RMC5RMC3RCXCR4CHRM2
SCHEMBL10483999 0.93 MC4R (0.47) MC4RMC5RMC3RCXCR4CHRM2
SCHEMBL10483864 0.81 SIGMAR1 (0.47) HDAC1CYP11B1CYP11B2NOS1
SCHEMBL7996321 0.80 CHRM2 (0.43) CXCR4CHRM2HDAC1CYP11B1CYP11B2
SCHEMBL5884099 0.80 MC4R (0.42) MC4RMC5RMC3RCXCR4CHRM2
SCHEMBL5884859 0.80 KDM4E (0.50) MC4RMC5RMC3RCHRM2HDAC1
SCHEMBL7981951 0.79 CXCR4 (0.38) CXCR4CHRM2HDAC1CYP11B1CYP11B2
SCHEMBL10863389 0.77 MC4R (0.46) MC4RMC5RMC3RCXCR4CHRM2
SCHEMBL23124232 0.77 CYP2A6 (0.48) CYP11B1CYP11B2MAOBCYP3A4
SCHEMBL7995384 0.77 MC4R (0.41) MC4RMC5RMC3RCXCR4CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39140-E1 Heterocyclic compounds BAYER CROPSCIENCE K.K. (JP) 2006-06-20 US disclosed
US-RE39129-E1 Heterocyclic compounds BAYER CROPSCIENCE K.K. (JP) 2006-06-13 US disclosed