SCHEMBL5885689

SCHEMBL5885689

Cc1cc(C#CCN(Cc2ccccc2)c2cccc(C#N)c2)ccc1C(=O)C(C)C

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGES O14684 9/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
KMT2A Q03164 1/20 0.40
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
NR3C1 P04150 1/20 0.39
FFAR1 O14842 1/20 0.38
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
TMEM97 Q5BJF2 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36
GFER P55789 1/20 0.36
KCNN4 O15554 1/20 0.35
KCNA5 P22460 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5885457 0.88 MEN1 (0.43) PTGESMEN1NPC1KMT2ACRHBP
SCHEMBL5885640 0.85 PTPN1 (0.37) PTGESKMT2ACRHBPCRHR2
SCHEMBL5885273 0.84 PPARG (0.40) KMT2AFFAR1MRGPRX4GFERKCNN4
SCHEMBL5886153 0.84 AR (0.48) PTGESMEN1NPC1KMT2ACRHBP
Hydrochloric Acid SCHEMBL5886012 0.84 PTPN1 (0.37) PTGESKMT2ACRHBPCRHR2
SCHEMBL5885776 0.84 KDM1A (0.39) PTGESMEN1NPC1KMT2ACRHBP
SCHEMBL5885627 0.75 PDK1 (0.40) PTGES
SCHEMBL5885884 0.74 PTPN1 (0.39) PTGESKMT2ACRHBPCRHR2NR3C1
SCHEMBL5885843 0.74 ACACB (0.41) NPC1MRGPRX4
Hydrochloric Acid SCHEMBL5885907 0.73 PTPN1 (0.39) PTGESKMT2ACRHBPCRHR2NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7005437-B2 Substituted aryl and heteroaryl derivatives, the preparation thereof and the use therof as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA KG (DE) 2006-02-28 US disclosed
US-20030045712-A1 Substituted aryl and heteroaryl derivatives, the preparation thereof and the use therof as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA KG (DE) 2003-03-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030045712-A1 Substituted aryl and heteroaryl derivatives, the preparation thereof and the use therof as pharmaceutical compositions F2, F12, F3 PTGES 2138/4885MEN1 1171/4885NPC1 2909/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.