SCHEMBL5886587

SCHEMBL5886587

c1cc(C2CCC2)ccc1C1CCC1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 13/20 0.56
ESR1 P03372 5/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
HDAC1 Q13547 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
POLB P06746 1/20 0.43
NOTUM Q6P988 1/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
HSP90AA1 P07900 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5148273 0.97 ESR2 (0.60) ESR2ESR1CYP3A4CYP2D6CYP2C9
SCHEMBL781509 0.93 HDAC1 (0.54) ESR2ESR1CYP3A4CYP2D6CYP2C9
SCHEMBL6275125 0.90 HDAC8 (0.52) ESR2HDAC1HDAC8HDAC6NOTUM
SCHEMBL28584923 0.90 HDAC8 (0.52) ESR2HDAC1HDAC8HDAC6NOTUM
SCHEMBL15260520 0.90 HDAC8 (0.52) ESR2HDAC1HDAC8HDAC6NOTUM
SCHEMBL5147779 0.90 ESR2 (0.54) ESR2ESR1CYP3A4CYP2D6CYP2C9
SCHEMBL42782 0.90 HDAC8 (0.52) ESR2HDAC1HDAC8HDAC6NOTUM
SCHEMBL5146632 0.87 ESR2 (0.52) ESR2ESR1CYP3A4CYP2D6CYP2C9
SCHEMBL25253951 0.86 ESR2 (0.47) ESR2ESR1CYP3A4CYP2D6CYP2C9
SCHEMBL435619 0.86 HTR3A (0.59) ESR2ESR1CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7138554-B2 Synthesis of (dibromocyclobuta) aromatic compounds TECHNION RESEARCH AND DEVELOPMENT FOUNDATION (IL) 2006-11-21 US disclosed
JP-2005132735-A POLYFUNCTIONAL CYCLOBUTABENZENE AND METHOD FOR PRODUCING THE SAME JAPAN SCIENCE & TECHNOLOGY AGENCY 2005-05-26 JP disclosed
US-20040116755-A1 Synthesis of (Dibromocyclobuta) aromatic compounds TECHNION RESEARCH AND DEVELOPMENT FOUNDATION (IL) 2004-06-17 US disclosed
WO-2002102810-A2 SYNTHESIS OF (DIBROMOCYCLOBUTA) AROMATIC COMPOUNDS TECHNION RESEARCH AND DEVELOPMENT FOUNDATION LTD. (IL) 2002-12-27 WO disclosed
US-5770763-A POLYARYLCYCLOBUTENES DERIVED FROM 3,6 FUNCTIONALIZED MONO AND DICYCLOBUTABENZENE THE BOARD OF REGENTS OF THE UNIV. OF MICHIGAN (US) 1998-06-23 US disclosed
US-5552508-A Difunctional bitricyclodecatriene monomers UNIVERSITY OF MICHIGAN, THE BOARD OF REGENTS (US) 1996-09-03 US disclosed