SCHEMBL5886967

SCHEMBL5886967

Cc1nc[nH]c2nc(=O)ccc1-2

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
PDPK1 O15530 1/20 0.33
PARP1 P09874 4/20 0.33
PIM1 P11309 2/20 0.33
CHEK1 O14757 1/20 0.33
RPS6KA3 P51812 1/20 0.33
KDM5B Q9UGL1 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
GAA P10253 1/20 0.30
ACVR1 Q04771 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8805425 0.73 ALDH1A1 (0.37) PDE3BPDE3APARP1ALDH1A1POLB
SCHEMBL17268292 0.72 VHL (0.40) PDE3BPDE3AGAA
SCHEMBL17298928 0.63 DCUN1D1 (0.46) ALDH1A1GAAHTT
Hydrochloric Acid SCHEMBL6225223 0.61 IDO1 (0.40) ALDH1A1POLBMAPT
SCHEMBL8404474 0.61
SCHEMBL20844021 0.60
SCHEMBL677524 0.59
SCHEMBL503673 0.58
SCHEMBL19493860 0.58
SCHEMBL17773604 0.58

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed