SCHEMBL5887552

SCHEMBL5887552

Cc1ccc(COC2=CC[CH]C=C2OC2CCCC2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.35
HRH3 Q9Y5N1 1/20 0.35
DRD4 P21917 2/20 0.33
TMEM97 Q5BJF2 2/20 0.33
SIGMAR1 Q99720 2/20 0.33
C5AR1 P21730 1/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KDM4E B2RXH2 1/20 0.33
CASP3 P42574 1/20 0.33
SENP8 Q96LD8 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
SENP6 Q9GZR1 1/20 0.33
AGXT P21549 2/20 0.33
MAOA P21397 3/20 0.32
ALDH1A1 P00352 2/20 0.32
NAAA Q02083 1/20 0.32
KMT2A Q03164 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874456 0.74 PDE4A (0.36) KMT2A
SCHEMBL6047662 0.73 SLC6A4 (0.34) KMT2A
SCHEMBL5907513 0.72 AGXT (0.36) MAOBHRH3NPC1RAB9ASMN1; SMN2
SCHEMBL18615830 0.68 NAAA (0.51) DRD4TMEM97SIGMAR1KDM4EAGXT
SCHEMBL11587452 0.67 NAAA (0.54) HRH3DRD4TMEM97SIGMAR1NPC1
SCHEMBL18616195 0.64 NAAA (0.59) HRH3DRD4TMEM97SIGMAR1AGXT
SCHEMBL8171032 0.62 EGFR (0.49) MAOBHRH3KDM4EALDH1A1KMT2A
SCHEMBL257928 0.61 EGFR (0.48) MAOBHRH3KDM4EALDH1A1KMT2A
SCHEMBL16979035 0.61 NAAA (0.54) HRH3DRD4TMEM97SIGMAR1AGXT
SCHEMBL8930166 0.61 NAAA (0.54) HRH3DRD4TMEM97SIGMAR1AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037931-B2 Corticotropin releasing factor moderator; analgesics; drug abruse, drug dependency; schizophrenia JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-02 US claimed
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed