SCHEMBL589534

SCHEMBL589534

CC(C)Oc1cc(Nc2cc(OC(CO)CO)nc(NC(C)c3ccc(F)cn3)n2)n[nH]1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 12/20 0.57
JAK2 O60674 8/20 0.47
JAK3 P52333 7/20 0.47
AURKA O14965 5/20 0.47
IGF1R P08069 3/20 0.47
FLT3 P36888 3/20 0.47
NTRK3 Q16288 2/20 0.47
NTRK2 Q16620 2/20 0.47
FGFR1 P11362 2/20 0.47
PTK2 Q05397 2/20 0.47
BTK Q06187 2/20 0.47
ALK Q9UM73 2/20 0.47
KCNH2 Q12809 2/20 0.47
LCK P06239 2/20 0.47
RET P07949 2/20 0.47
FYN P06241 1/20 0.47
FLT1 P17948 1/20 0.47
LTK P29376 1/20 0.47
KDR P35968 1/20 0.47
CSNK1A1 P48729 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL589533 1.00 NTRK1 (0.57) NTRK1JAK2JAK3AURKAIGF1R
SCHEMBL589089 0.86 NTRK1 (0.65) NTRK1JAK2JAK3AURKAIGF1R
SCHEMBL589432 0.84 NTRK1 (0.76) NTRK1JAK2JAK3AURKAIGF1R
SCHEMBL589431 0.84 NTRK1 (0.76) NTRK1JAK2JAK3AURKAIGF1R
SCHEMBL588554 0.80 NTRK1 (0.60) NTRK1JAK2JAK3AURKAIGF1R
SCHEMBL588553 0.80 NTRK1 (0.60) NTRK1JAK2JAK3AURKAIGF1R
SCHEMBL588638 0.79 NTRK1 (0.55) NTRK1JAK2JAK3AURKAIGF1R
SCHEMBL588783 0.78 JAK3 (0.57) NTRK1JAK2JAK3AURKAIGF1R
SCHEMBL3041951 0.78 NTRK1 (0.69) NTRK1JAK2JAK3AURKAIGF1R
SCHEMBL589107 0.78 NTRK1 (0.77) NTRK1JAK2JAK3AURKAIGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8114989-B2 Pyrazolylaminopyrimidine derivatives useful as tyrosine kinase inhibitors ASTRAZENECA AB (SE) 2012-02-14 US claimed