SCHEMBL5897233

SCHEMBL5897233

Cc1ccc(NC(=O)c2cccc(N(C)C)c2)cc1NC(=O)c1cc2cccnc2nc1C

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 12/20 0.61
BRAF P15056 4/20 0.61
KDM4E B2RXH2 2/20 0.61
ALDH1A1 P00352 2/20 0.61
MAPT P10636 2/20 0.61
HPGD P15428 2/20 0.61
RAF1 P04049 1/20 0.61
TP53 P04637 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61
CYP2C9 P11712 1/20 0.61
ALOX15 P16050 1/20 0.61
MAPK11 Q15759 1/20 0.61
HSD17B10 Q99714 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61
CSF1R P07333 2/20 0.59
SMO Q99835 2/20 0.58
SIRT1 Q96EB6 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5897487 0.84 CSF1R (0.81) MAPK14BRAFKDM4EALDH1A1MAPT
SCHEMBL6484862 0.79 MAPK14 (0.85) MAPK14BRAFKDM4EALDH1A1MAPT
SCHEMBL6477991 0.78 MAPK14 (0.76) MAPK14BRAFKDM4EALDH1A1MAPT
SCHEMBL5007830 0.78 MAPK14 (0.72) MAPK14BRAFKDM4EALDH1A1MAPT
SCHEMBL6477729 0.78 MAPK14 (0.74) MAPK14BRAFKDM4EALDH1A1MAPT
SCHEMBL2978412 0.77 CSF1R (0.70) MAPK14BRAFKDM4EALDH1A1MAPT
SCHEMBL10028403 0.77 MAPK14 (0.85) MAPK14BRAFKDM4EALDH1A1MAPT
SCHEMBL6477982 0.77 MAPK14 (0.70) MAPK14BRAFKDM4EALDH1A1MAPT
SCHEMBL6781525 0.76 MAPK14 (0.83) MAPK14BRAFKDM4EALDH1A1MAPT
SCHEMBL1424183 0.76 MAPK14 (1.00) MAPK14BRAFKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060700-B2 Amide derivatives useful as inhibitors of the production of cytokines ASTRAZENECA AB (SE) 2006-06-13 US disclosed
US-20030105142-A1 Amide derivatives useful as inhibitors of the production of cytokines ASTRAZENECA AB 2003-06-05 US disclosed
US-6432949-B1 Amide derivatives useful as inhibitors of the production of cytokines ASTRAZENECA AB (SE) 2002-08-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030105142-A1 Amide derivatives useful as inhibitors of the production of cytokines IL6, IL6ST, IL2 MAPK14 2563/4885BRAF 1764/4885KDM4E 1955/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.