SCHEMBL5899698

SCHEMBL5899698

COCCOC(=O)N1CCC(C#N)(NC(=O)C(CC(C)C)OC(=O)NCc2ccccc2)C1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSL P07711 11/20 0.41
CTSS P25774 7/20 0.38
CTSK P43235 5/20 0.38
CTSB P07858 4/20 0.38
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3895283 0.95 CTSL (0.39) CTSLCTSSCTSKCTSBJAK2
SCHEMBL3898963 0.92 CTSL (0.43) CTSLCTSSCTSKCTSBALDH1A1
SCHEMBL3896939 0.91 CTSL (0.42) CTSLCTSSCTSKCTSB
SCHEMBL3898205 0.88 CTSL (0.45) CTSLCTSSCTSKCTSB
SCHEMBL3894998 0.87 CTSL (0.46) CTSLCTSSCTSKCTSBALDH1A1
SCHEMBL3900293 0.87 CTSL (0.44) CTSLCTSSCTSKCTSB
SCHEMBL3903294 0.86 CTSL (0.46) CTSLCTSSCTSKCTSB
SCHEMBL3899281 0.85 CTSL (0.43) CTSLCTSSCTSKCTSB
SCHEMBL7482961 0.85 CTSL (0.49) CTSLCTSSCTSKCTSB
SCHEMBL3910469 0.85 CTSL (0.42) CTSLCTSSCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6982263-B2 Nitriles useful as reversible inhibitors of cysteine proteases BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2006-01-03 US claimed