SCHEMBL5915925

SCHEMBL5915925

Cc1c(O)ccnc1-c1ccc2[nH]nc(C(=O)Nc3ccncc3)c2c1.N#Cc1cccc(NC(=O)c2n[nH]c3ccc(-c4cnco4)cc23)c1

nearest known ligand 0.53

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 20/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL82445 0.86 LRRK2 (0.56) LRRK2
SCHEMBL4523534 0.83 DYRK1A (0.53) LRRK2
SCHEMBL81160 0.82 DYRK1A (0.54) LRRK2
SCHEMBL952067 0.79 DYRK1A (0.55) LRRK2
SCHEMBL4519531 0.71 LRRK2 (0.57) LRRK2
Hydrochloric Acid SCHEMBL4523142 0.70 LRRK2 (0.56) LRRK2
SCHEMBL82789 0.70 DYRK1A (0.52) LRRK2
SCHEMBL5945615 0.70 FLT3 (0.60)
SCHEMBL22890140 0.70 LRRK2 (1.00) LRRK2
SCHEMBL29771523 0.70 LRRK2 (1.00) LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060004000-A1 Indazolecarboxamide derivatives, preparation and use thereof as CDK1, CDK2 and CDK4 inhibitors SANOFI-AVENTIS (FR) 2006-01-05 US claimed
US-20060004000-A1 Indazolecarboxamide derivatives, preparation and use thereof as CDK1, CDK2 and CDK4 inhibitors SANOFI-AVENTIS (FR) 2006-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060004000-A1 Indazolecarboxamide derivatives, preparation and use thereof as CDK1, CDK2 and CDK4 inhibitors CDK2, CDK1, CDK4 LRRK2 1183/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.