SCHEMBL5951455

SCHEMBL5951455

CCCCC=Cc1cccc2c1C(=O)C(C)C2

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACHE P22303 6/20 0.40
ABCB1 P08183 1/20 0.36
PDE5A O76074 1/20 0.35
MAOA P21397 2/20 0.35
MAOB P27338 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
CYSLTR2 Q9NS75 2/20 0.33
CYSLTR1 Q9Y271 2/20 0.33
IAPP P10997 1/20 0.33
BID P55957 3/20 0.32
BCL2L1 Q07817 3/20 0.32
MCL1 Q07820 3/20 0.32
BAK1 Q16611 3/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
FAAH O00519 1/20 0.31
MGLL Q99685 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5951451 1.00 ACHE (0.40) ACHEABCB1PDE5AMAOAMAOB
SCHEMBL5951520 0.80 ACHE (0.49) ACHEPDE5AL3MBTL1CYSLTR2CYSLTR1
SCHEMBL5951524 0.80 ACHE (0.49) ACHEPDE5AL3MBTL1CYSLTR2CYSLTR1
SCHEMBL5951538 0.76 ACHE (0.42) ACHEABCB1MAOAMAOB
SCHEMBL5951674 0.76 ACHE (0.46) ACHEABCB1MAOAMAOB
SCHEMBL5953058 0.76 ACHE (0.46) ACHEABCB1MAOAMAOB
SCHEMBL5951542 0.76 ACHE (0.42) ACHEABCB1MAOAMAOB
SCHEMBL5952113 0.74 ACHE (0.44) ACHEABCB1MAOAMAOBBID
SCHEMBL5951816 0.74 ACHE (0.41) ACHEABCB1MAOAMAOB
SCHEMBL5951540 0.71 ACHE (0.41) ACHEABCB1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7038070-B2 Preparation of preparing substituted indanones BASELL POLYOLEFINE GMBH (DE) 2006-05-02 US disclosed
US-6963017-B2 Preparation of preparing substituted indanones BASELL POLYOLEFINE GMBH (DE) 2005-11-08 US disclosed
EP-0968158-B1 METHOD OF PREPARING SUBSTITUTED INDANONES, THE SUBSTITUTED INDANONES AND METALLOCENES PREPARED THEREFROM BASELL POLYOLEFINE GMBH (DE) 2005-08-10 EP disclosed
US-20050033076-A1 Preparation of preparing substituted indanones EQUISTAR CHEMICALS, LP 2005-02-10 US disclosed
US-20030009046-A1 Preparation of preparing substituted indanones EQUISTAR CHEMICALS, LP 2003-01-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050033076-A1 Preparation of preparing substituted indanones CYP1A2, CYP2J2, IDH3A ACHE 839/4885ABCB1 1146/4885PDE5A 2758/4885
US-20030009046-A1 Preparation of preparing substituted indanones CYP1A2, CYP1B1, CYP1A1 ACHE 820/4885ABCB1 1132/4885PDE5A 2954/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.