SCHEMBL5959631

SCHEMBL5959631

Clc1ccsc1-c1nc(-c2cccc(CBr)c2Cl)no1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 15/20 0.55
ABCG2 Q9UNQ0 1/20 0.38
GRM5 P41594 1/20 0.36
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPK1 P28482 1/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4587506 0.81 CASP3 (0.68) CASP3GRM5RAB9A
SCHEMBL4587239 0.77 CASP3 (0.72) CASP3SMN1; SMN2
SCHEMBL4552076 0.72 CASP3 (1.00) CASP3NPC1RAB9ATDP1MAPK1
SCHEMBL4415506 0.72 CASP3 (0.68) CASP3GRM5NPC1RAB9ASMN1; SMN2
SCHEMBL4552769 0.71 CASP3 (0.78) CASP3GRM5
SCHEMBL4586852 0.71 CASP3 (0.67) CASP3NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL4593616 0.70 CASP3 (0.62) CASP3NPC1RAB9ASMN1; SMN2TDP1
SCHEMBL4586808 0.69 CASP3 (0.69) CASP3GRM5
SCHEMBL4552210 0.69 CASP3 (1.00) CASP3NPC1RAB9ASMN1; SMN2L3MBTL1
SCHEMBL4587234 0.69 CASP3 (0.63) CASP3NPC1RAB9ASMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7144876-B2 3,5-Disubstituted-[1,2,4]-oxadiazoles and analogs as activators of caspases and inducers of apoptosis and the use thereof CYTOVIA, INC. (US) 2006-12-05 US claimed