SCHEMBL5960477

SCHEMBL5960477

CC(=O)Nc1nc(C)c(-c2csc([AsH2])n2)s1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 7/20 0.73
PIK3CD O00329 1/20 0.68
PIK3CA P42336 1/20 0.68
PIK3CB P42338 1/20 0.68
MEN1 O00255 2/20 0.67
KMT2A Q03164 2/20 0.67
POLB P06746 1/20 0.67
PI4KB Q9UBF8 5/20 0.65
KDM4E B2RXH2 2/20 0.63
ALDH1A1 P00352 2/20 0.63
MAPT P10636 2/20 0.63
HTT P42858 2/20 0.63
HSD17B10 Q99714 2/20 0.63
USP2 O75604 1/20 0.63
LMNA P02545 1/20 0.63
GAA P10253 1/20 0.63
ALOX15 P16050 1/20 0.63
TSHR P16473 1/20 0.63
GFER P55789 1/20 0.63
NPSR1 Q6W5P4 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4534987 0.84 PIK3CG (1.00) PIK3CGPIK3CDPIK3CAPIK3CBMEN1
SCHEMBL16882665 0.83 PIK3CG (0.73) PIK3CGPIK3CDPIK3CAPIK3CBMEN1
SCHEMBL2833123 0.82 PIK3CG (0.71) PIK3CGPIK3CDPIK3CAPIK3CBMEN1
SCHEMBL29089046 0.82 PIK3CG (0.74) PIK3CGPIK3CDPIK3CAPIK3CBMEN1
SCHEMBL3511005 0.81 PIK3CG (1.00) PIK3CGPIK3CDPIK3CAPIK3CBMEN1
SCHEMBL2836277 0.81 PIK3CG (0.70) PIK3CGPIK3CDPIK3CAPIK3CBMEN1
SCHEMBL2831536 0.81 PIK3CG (0.70) PIK3CGPIK3CDPIK3CAPIK3CBMEN1
SCHEMBL2837166 0.81 PIK3CG (0.74) PIK3CGPIK3CDPIK3CAPIK3CBMEN1
SCHEMBL4532662 0.81 PIK3CG (1.00) PIK3CGPIK3CDPIK3CAPIK3CBMEN1
SCHEMBL3513224 0.81 PIK3CG (0.70) PIK3CGPIK3CDPIK3CAPIK3CBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1709019-A2 THIAZOLE DERIVATIVES AND USE THEREOF Applied Research Systems ARS Holding N.V. (AN) 2006-10-11 EP disclosed
WO-2005068444-A2 THIAZOLE DERIVATIVES AND USE THEREOF APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2005-07-28 WO disclosed