SCHEMBL5968628

SCHEMBL5968628

CC(C)(Cc1cccc(C(=O)NCCCc2ccccc2)c1)NC[C@H](O)c1ccc(O)c(CO)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 16/20 0.68
ADRB1 P08588 5/20 0.61
CHRM3 P20309 1/20 0.59
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
TSHR P16473 2/20 0.49
ADRA1D P25100 2/20 0.49
KDM4E B2RXH2 2/20 0.49
HTR1A P08908 1/20 0.49
CHRM5 P08912 1/20 0.49
ADRB3 P13945 1/20 0.49
DRD2 P14416 1/20 0.49
ADRA2B P18089 1/20 0.49
DRD4 P21917 1/20 0.49
SLC6A2 P23975 1/20 0.49
FPR3 P25089 1/20 0.49
HTR1D P28221 1/20 0.49
HTR1B P28222 1/20 0.49
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5968634 1.00 ADRB2 (0.68) ADRB2ADRB1CHRM3CYP1A2CYP2D6
SCHEMBL5968865 0.95 ADRB2 (0.61) ADRB2ADRB1CHRM3CYP1A2CYP2D6
SCHEMBL5968861 0.95 ADRB2 (0.61) ADRB2ADRB1CHRM3CYP1A2CYP2D6
SCHEMBL5968883 0.95 ADRB2 (0.70) ADRB2ADRB1CHRM3CYP1A2CYP2D6
SCHEMBL5968882 0.95 ADRB2 (0.70) ADRB2ADRB1CHRM3CYP1A2CYP2D6
SCHEMBL5969116 0.93 ADRB2 (0.59) ADRB2ADRB1CHRM3CYP1A2CYP2D6
SCHEMBL5969113 0.93 ADRB2 (0.59) ADRB2ADRB1CHRM3CYP1A2CYP2D6
SCHEMBL5968667 0.91 ADRB2 (0.65) ADRB2ADRB1CHRM3CYP1A2CYP2D6
SCHEMBL5968672 0.91 ADRB2 (0.65) ADRB2ADRB1CHRM3CYP1A2CYP2D6
SCHEMBL5968881 0.90 ADRB2 (0.57) ADRB2ADRB1CHRM3CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1727789-A2 PHENYLETHANOLAMINE DERIVATIVES AS BETA-2 AGONISTS Pfizer Limited (GB) 2006-12-06 EP claimed
WO-2005090287-A2 PHENYLETHANOLAMINE DERIVATIVES AS BETA-2 AGONISTS PFIZER LIMITED (GB) 2005-09-29 WO claimed
EP-1727789-A2 PHENYLETHANOLAMINE DERIVATIVES AS BETA-2 AGONISTS Pfizer Limited (GB) 2006-12-06 EP disclosed
WO-2005090287-A2 PHENYLETHANOLAMINE DERIVATIVES AS BETA-2 AGONISTS PFIZER LIMITED (GB) 2005-09-29 WO disclosed