SCHEMBL5973802

SCHEMBL5973802

O=C(Cc1ccccc1)c1nc2ccccc2s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 1.00
SMN1; SMN2 Q16637 5/20 1.00
NPC1 O15118 4/20 1.00
HPGD P15428 3/20 1.00
ALDH1A1 P00352 4/20 0.72
MAPT P10636 3/20 0.72
GAA P10253 1/20 0.72
MCL1 Q07820 1/20 0.72
L3MBTL1 Q9Y468 3/20 0.62
NFKB1 P19838 2/20 0.58
NFKB2 Q00653 2/20 0.58
RELA Q04206 2/20 0.58
CSNK1D P48730 2/20 0.58
GLO1 Q04760 2/20 0.55
PKM P14618 1/20 0.55
HTR1A P08908 3/20 0.50
DRD2 P14416 2/20 0.50
SLC6A4 P31645 2/20 0.50
HTR7 P34969 2/20 0.50
TSHR P16473 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6179039 0.87 NPC1 (0.76) RAB9ASMN1; SMN2NPC1HPGDALDH1A1
SCHEMBL1667036 0.84 NPC1 (0.72) RAB9ASMN1; SMN2NPC1HPGDALDH1A1
Trifluoroacetic Acid SCHEMBL7452391 0.83 NPC1 (0.70) RAB9ASMN1; SMN2NPC1HPGDALDH1A1
SCHEMBL1950317 0.81 NPC1 (0.68) RAB9ASMN1; SMN2NPC1HPGDL3MBTL1
SCHEMBL2097484 0.80 RAB9A (0.67) RAB9ASMN1; SMN2NPC1HPGDALDH1A1
SCHEMBL6647582 0.80 RAB9A (0.67) RAB9ASMN1; SMN2NPC1HPGDALDH1A1
SCHEMBL16808929 0.80 RAB9A (0.67) RAB9ASMN1; SMN2NPC1HPGDALDH1A1
SCHEMBL10313749 0.80 RAB9A (0.67) RAB9ASMN1; SMN2NPC1HPGDALDH1A1
SCHEMBL27394846 0.80 NPC1 (0.65) RAB9ASMN1; SMN2NPC1HPGDALDH1A1
SCHEMBL28727291 0.79 SMN1; SMN2 (0.65) RAB9ASMN1; SMN2NPC1HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1007514-B1 HETEROCYCLIC KETONES AS NPY Y5 ANTAGONISTS BAYER CORP (US) 2006-11-15 EP disclosed
EP-1007514-A1 HETEROCYCLIC KETONES AS NPY Y5 ANTAGONISTS Bayer Corporation (US) 2000-06-14 EP disclosed
WO-1999010330-A1 HETEROCYCLIC KETONES AS NPY Y5 ANTAGONISTS BAYER CORPORATION (US) 1999-03-04 WO disclosed