Almestrone

Almestrone

SCHEMBL5983577

CC1Cc2cc(O)ccc2[C@H]2CC[C@]3(C)C(=O)CC[C@H]3[C@H]12

nearest known ligand 0.65

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 11/20 0.65
HSD17B1 P14061 4/20 0.65
ESR1 P03372 3/20 0.65
STS P08842 2/20 0.65
ESR2 Q92731 2/20 0.65
LMNA P02545 2/20 0.65
SHBG P04278 2/20 0.65
CYP3A4 P08684 2/20 0.65
MAPT P10636 2/20 0.65
AKR1B10 O60218 1/20 0.65
CYP1A2 P05177 1/20 0.65
PGR P06401 1/20 0.65
SERPINA6 P08185 1/20 0.65
AR P10275 1/20 0.65
AKR1B1 P15121 1/20 0.65
NFKB1 P19838 1/20 0.65
SLC6A4 P31645 1/20 0.65
OPRM1 P35372 1/20 0.65
SNCA P37840 1/20 0.65
HTR2B P41595 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Almestrone SCHEMBL8089798 1.00 CYP19A1 (0.65) CYP19A1HSD17B1ESR1STSESR2
Almestrone SCHEMBL1657631 1.00 CYP19A1 (0.65) CYP19A1HSD17B1ESR1STSESR2
Almestrone SCHEMBL12364346 1.00 CYP19A1 (0.65) CYP19A1HSD17B1ESR1STSESR2
Almestrone SCHEMBL13216952 1.00 CYP19A1 (0.65) CYP19A1HSD17B1ESR1STSESR2
Almestrone SCHEMBL12364585 1.00 CYP19A1 (0.65) CYP19A1HSD17B1ESR1STSESR2
Almestrone SCHEMBL2244882 0.97 CYP19A1 (0.61) CYP19A1HSD17B1ESR1STSESR2
SCHEMBL8376406 0.88 CYP19A1 (0.65) CYP19A1HSD17B1ESR1STSESR2
SCHEMBL10083670 0.88 CYP19A1 (0.65) CYP19A1HSD17B1ESR1STSESR2
SCHEMBL10083683 0.88 CYP19A1 (0.65) CYP19A1HSD17B1ESR1STSESR2
SCHEMBL6879791 0.88 CYP19A1 (0.65) CYP19A1HSD17B1ESR1STSESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658306-A1 DELTA 15 -D-HOMOSTEROIDS HAVING AN ANDROGENIC EFFECT Schering AG (DE) 2006-05-24 EP disclosed
WO-2005021573-A1 Δ15-D-HOMOSTEROIDS HAVING AN ANDROGENIC EFFECT SCHERING AG (DE) 2005-03-10 WO disclosed
US-3929844-A 3-Cyclopentyl ethers of 7{60 -methyl estrone CIBA GEIGY CORP 1975-12-30 US disclosed