SCHEMBL5988086

SCHEMBL5988086

O=C1Nc2ccncc2C1=Cc1sccc1Br

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.68
MAPT P10636 2/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
RAF1 P04049 3/20 0.41
PIK3C3 Q8NEB9 1/20 0.41
TLK2 Q86UE8 2/20 0.38
CDK5 Q00535 1/20 0.38
PTK2B Q14289 1/20 0.38
CDK5R1 Q15078 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAP1LC3B Q9GZQ8 1/20 0.37
GSK3B P49841 2/20 0.37
TGM2 P21980 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5988992 0.90 KDR (0.68) KDRMAPTMAPK1HTTRAF1
SCHEMBL31060741 0.81 KDR (1.00) KDRMAPTHTTRAF1TLK2
SCHEMBL6001467 0.81 KDR (1.00) KDRMAPTHTTRAF1TLK2
SCHEMBL5988782 0.78 KDR (0.47) KDRMAPTMAPK1HTTTLK2
SCHEMBL5990000 0.76 PDPK1 (0.53) KDRMAPTMAPK1HTTTLK2
SCHEMBL5988900 0.74 KDR (0.64) KDRMAPTMAPK1HTTRAF1
SCHEMBL5988173 0.73 RET (0.43) KDRMAPTMAPK1HTTTLK2
SCHEMBL5374098 0.72 KDR (0.61) KDRMAPTMAPK1HTTRAF1
SCHEMBL5988934 0.72 KDR (0.54) KDRMAPTRAF1
SCHEMBL5988962 0.72 KDR (0.54) KDRMAPTMAPK1RAF1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849641-B1 Azaindole tyrosine kinase inhibitors SUGEN, INC. (US) 2005-02-01 US claimed
US-6987113-B2 Tyrosine kinase inhibitors SUGEN, INC. (US) 2006-01-17 US disclosed