SCHEMBL5995073

SCHEMBL5995073

CC(c1ccc(Cl)cc1)c1c(Cl)cc(-n2ncc(=O)[nH]c2=O)cc1Cl

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.69
NR1I2 O75469 1/20 0.69
KMT2A Q03164 1/20 0.69
THRB P10828 13/20 0.49
THRA P10827 4/20 0.49
P2RX7 Q99572 5/20 0.43
NPBWR1 P48145 1/20 0.40
MCHR1 Q99705 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6342801 0.86 MEN1 (0.71) MEN1NR1I2KMT2ATHRBTHRA
SCHEMBL5562109 0.85 MEN1 (0.69) MEN1NR1I2KMT2ATHRBTHRA
SCHEMBL10419955 0.83 MEN1 (0.64) MEN1NR1I2KMT2ATHRBTHRA
SCHEMBL10394519 0.83 MEN1 (0.64) MEN1NR1I2KMT2ATHRBTHRA
SCHEMBL5567070 0.82 MEN1 (0.60) MEN1NR1I2KMT2ATHRBTHRA
SCHEMBL6345637 0.82 MEN1 (0.65) MEN1NR1I2KMT2ATHRBTHRA
SCHEMBL5566905 0.82 MEN1 (0.65) MEN1NR1I2KMT2ATHRBTHRA
SCHEMBL9823772 0.82 MEN1 (0.65) MEN1NR1I2KMT2ATHRBTHRA
Diclazuril SCHEMBL126138 0.82 MEN1 (1.00) MEN1NR1I2KMT2ATHRBTHRA
SCHEMBL5566019 0.81 MEN1 (0.64) MEN1NR1I2KMT2ATHRBTHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012065139-A2 ENTPD5 INHIBITORS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-05-18 WO disclosed