SCHEMBL6004074

SCHEMBL6004074

CCCC(=O)Nc1cccn([C@@H](CC)C(=O)NC(CC(=O)O)C(=O)COc2c(F)c(F)cc(F)c2F)c1=O

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 11/20 0.59
CASP3 P42574 9/20 0.53
CASP6 P55212 7/20 0.53
CASP8 Q14790 7/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473185 1.00 CASP1 (0.59) CASP1CASP3CASP6CASP8
SCHEMBL2003067 1.00 CASP1 (0.59) CASP1CASP3CASP6CASP8
SCHEMBL2003069 1.00 CASP1 (0.59) CASP1CASP3CASP6CASP8
SCHEMBL473098 0.94 CASP1 (0.61) CASP1CASP3CASP6CASP8
SCHEMBL2003509 0.94 CASP1 (0.61) CASP1CASP3CASP6CASP8
SCHEMBL2003507 0.94 CASP1 (0.61) CASP1CASP3CASP6CASP8
SCHEMBL473113 0.92 CASP1 (0.59) CASP1CASP3CASP6CASP8
SCHEMBL473109 0.92 CASP1 (0.59) CASP1CASP3CASP6CASP8
SCHEMBL473111 0.92 CASP1 (0.59) CASP1CASP3CASP6CASP8
SCHEMBL6005359 0.91 CASP1 (0.61) CASP1CASP3CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1631549-A2 3-[2-(3-AMINO-2-OXO-2H-PYRIDIN-1-YL)-ACETYLAMINO]-4-OXO-PENTANOIC ACID DERIVATIVES AND THEIR USE AS CASPASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2006-03-08 EP disclosed
WO-2004106304-A2 3 - [2- (3-AMINO-2-OXO-2H-PYRIDIN-1-YL) - ACETYLAMINO] - 4- OXO-PENTANOIC ACID DERIVATIVES AND THEIR USE AS CASPASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2004-12-09 WO disclosed