SCHEMBL6004291

SCHEMBL6004291

Cc1sc2[nH]cnc(=O)c2c1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.54
BCAT2 O15382 1/20 0.37
MAPK1 P28482 2/20 0.36
LMNA P02545 2/20 0.36
ALDH1A1 P00352 2/20 0.36
USP2 O75604 1/20 0.36
HTT P42858 1/20 0.36
HPGD P15428 2/20 0.35
KDM4E B2RXH2 2/20 0.33
GAA P10253 1/20 0.33
QPCT Q16769 1/20 0.33
LIMK1 P53667 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CDC7 O00311 1/20 0.33
ROCK2 O75116 1/20 0.33
MAP4K4 O95819 1/20 0.33
PIM1 P11309 1/20 0.33
GSK3B P49841 1/20 0.33
HIPK2 Q9H2X6 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30987690 0.78 BCAT2 (0.60) PDPK1BCAT2LMNAALDH1A1HTT
SCHEMBL9595093 0.78 PDPK1 (0.46) PDPK1BCAT2MAPK1LMNAALDH1A1
SCHEMBL30987724 0.77 BCAT2 (0.44) PDPK1BCAT2LMNAALDH1A1HTT
SCHEMBL9852516 0.70 PDPK1 (0.46) PDPK1ALDH1A1GAAMEN1KMT2A
SCHEMBL12102045 0.69 MAPK1 (0.55) PDPK1MAPK1LMNAALDH1A1HTT
SCHEMBL8404455 0.66
SCHEMBL1101927 0.63 MAPK1 (0.44) MAPK1ALDH1A1HTTHPGDKDM4E
SCHEMBL11579887 0.62 CSNK2A1 (0.57) PDPK1BCAT2ALDH1A1HTTHPGD
SCHEMBL6239318 0.62 PIM1 (0.37) PDPK1LMNAALDH1A1HTTHPGD
SCHEMBL3036602 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed
US-5254679-A Containing a quaternized nitrogen IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-10-19 US disclosed
EP-0164944-B1 CEPHALOSPORIN DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-07-11 EP disclosed
EP-0164944-A1 Cephalosporin derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-12-18 EP disclosed