SCHEMBL6004373

SCHEMBL6004373

COc1cc2nccc(Oc3ccc(C)nc3-c3ncccn3)c2cc1OC

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 1/20 0.55
PDGFRA P16234 1/20 0.55
SRC P12931 5/20 0.53
TGFBR1 P36897 5/20 0.53
EGFR P00533 1/20 0.50
FGFR2 P21802 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3906631 0.87 TGFBR1 (0.53) PDGFRBPDGFRASRCTGFBR1EGFR
SCHEMBL3897952 0.87 FGFR2 (0.56) PDGFRBPDGFRASRCTGFBR1EGFR
SCHEMBL4487210 0.86 PDGFRB (0.53) PDGFRBPDGFRASRCTGFBR1EGFR
SCHEMBL3891418 0.86 SRC (0.55) PDGFRBPDGFRASRCTGFBR1EGFR
SCHEMBL3906510 0.85 SRC (0.53) PDGFRBPDGFRASRCTGFBR1EGFR
SCHEMBL6005275 0.85 PDGFRB (0.52) PDGFRBPDGFRASRCTGFBR1EGFR
SCHEMBL3897482 0.84 SRC (0.55) PDGFRBPDGFRASRCTGFBR1EGFR
SCHEMBL3894826 0.84 PDGFRB (0.54) PDGFRBPDGFRASRCTGFBR1EGFR
SCHEMBL3893874 0.84 SRC (0.57) PDGFRBPDGFRASRCTGFBR1FGFR2
SCHEMBL3905667 0.84 PDGFRA (0.51) PDGFRBPDGFRASRCTGFBR1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed