SCHEMBL6004614

SCHEMBL6004614

COC(=O)c1ccc(NC=C2C(=O)OC(C)(C)OC2=O)cc1Cl

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 18/20 0.55
HSD17B10 Q99714 3/20 0.55
MAPK1 P28482 1/20 0.55
CYP1A2 P05177 2/20 0.54
CYP3A4 P08684 2/20 0.54
RAB9A P51151 1/20 0.54
TSHR P16473 1/20 0.51
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
KDM4E B2RXH2 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.43
NPSR1 Q6W5P4 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30905509 0.89 ALDH1A1 (0.59) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL30905503 0.89 ALDH1A1 (0.59) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL1890105 0.86 ALDH1A1 (0.59) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL22766451 0.85 ALDH1A1 (0.55) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL21200929 0.85 ALDH1A1 (0.58) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL6004820 0.85 ALDH1A1 (0.58) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL21200952 0.84 ALDH1A1 (0.56) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL30616279 0.83 ALDH1A1 (0.59) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL2174228 0.83 ALDH1A1 (0.59) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4
SCHEMBL27402291 0.81 ALDH1A1 (0.51) ALDH1A1HSD17B10MAPK1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed