SCHEMBL6005322

SCHEMBL6005322

CCCS(=O)(=O)Nc1cccn([C@@H](CC)C(=O)NC(CC(=O)O)C(=O)COc2c(F)c(F)cc(F)c2F)c1=O

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 3/20 0.54
CASP3 P42574 17/20 0.50
CASP6 P55212 16/20 0.50
CASP8 Q14790 16/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473275 1.00 CASP1 (0.54) CASP1CASP3CASP6CASP8
SCHEMBL473276 1.00 CASP1 (0.54) CASP1CASP3CASP6CASP8
SCHEMBL473274 1.00 CASP1 (0.54) CASP1CASP3CASP6CASP8
SCHEMBL2001699 0.95 CASP1 (0.56) CASP1CASP3CASP6CASP8
SCHEMBL2001700 0.95 CASP1 (0.56) CASP1CASP3CASP6CASP8
SCHEMBL473171 0.90 CASP1 (0.54) CASP1CASP3CASP6CASP8
SCHEMBL473172 0.90 CASP1 (0.54) CASP1CASP3CASP6CASP8
SCHEMBL473170 0.90 CASP1 (0.54) CASP1CASP3CASP6CASP8
SCHEMBL473217 0.89 CASP1 (0.55) CASP1CASP3CASP6CASP8
SCHEMBL473214 0.89 CASP1 (0.55) CASP1CASP3CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1631549-A2 3-[2-(3-AMINO-2-OXO-2H-PYRIDIN-1-YL)-ACETYLAMINO]-4-OXO-PENTANOIC ACID DERIVATIVES AND THEIR USE AS CASPASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2006-03-08 EP disclosed
WO-2004106304-A2 3 - [2- (3-AMINO-2-OXO-2H-PYRIDIN-1-YL) - ACETYLAMINO] - 4- OXO-PENTANOIC ACID DERIVATIVES AND THEIR USE AS CASPASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2004-12-09 WO disclosed