SCHEMBL6005536

SCHEMBL6005536

CCCCC1N(C)C(=O)OC12CCN(C1CCN(C(=O)c3cccc(C)c3C)CC1)CC2

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 13/20 0.65
HSD11B1 P28845 1/20 0.43
KMT2A Q03164 1/20 0.42
CHRM2 P08172 1/20 0.42
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
TP53BP1 Q12888 1/20 0.39
L3MBTL3 Q96JM7 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CHRM1 P11229 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6008613 0.87 CCR5 (0.71) CCR5
SCHEMBL6008994 0.87 CCR5 (0.69) CCR5
SCHEMBL6009109 0.86 CCR5 (0.88) CCR5HSD11B1KMT2ACHRM2
SCHEMBL6007364 0.86 CCR5 (0.61) CCR5TP53BP1L3MBTL3L3MBTL1
SCHEMBL6007031 0.85 CCR5 (0.60) CCR5KMT2ATP53BP1L3MBTL3L3MBTL1
SCHEMBL6008620 0.83 CCR5 (0.63) CCR5
SCHEMBL6009248 0.82 CCR5 (0.57) CCR5
SCHEMBL6008414 0.81 CCR5 (0.81) CCR5CHRM2
SCHEMBL6008456 0.81 CCR5 (0.81) CCR5CHRM2
SCHEMBL6009045 0.81 CCR5 (0.61) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716156-A2 CHEMOKINE CCR5 RECEPTOR MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2006-11-02 EP claimed
WO-2005075484-A2 CHEMOKINE CCR5 RECEPTOR MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-08-18 WO claimed