SCHEMBL6006576

SCHEMBL6006576

CCCCC1N(CC2CCCCC2)C(=O)OC12CCN(C1CCN(C(=O)c3ccncc3)CC1)CC2

nearest known ligand 0.75

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 16/20 0.75
KDM4E B2RXH2 1/20 0.44
OPRM1 P35372 1/20 0.40
OPRL1 P41146 1/20 0.40
MBTD1 Q05BQ5 2/20 0.40
L3MBTL3 Q96JM7 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6005547 0.92 CCR5 (0.81) CCR5KDM4EMBTD1L3MBTL3L3MBTL1
SCHEMBL6006847 0.91 CCR5 (0.73) CCR5
SCHEMBL6005860 0.89 CCR5 (0.78) CCR5
SCHEMBL6008091 0.89 CCR5 (0.73) CCR5MBTD1L3MBTL3L3MBTL1
SCHEMBL6008167 0.88 CCR5 (0.72) CCR5MBTD1L3MBTL3L3MBTL1
SCHEMBL6008381 0.88 CCR5 (0.72) CCR5
SCHEMBL6005538 0.87 CCR5 (0.76) CCR5MBTD1L3MBTL3L3MBTL1
SCHEMBL6009200 0.87 CCR5 (0.69) CCR5
SCHEMBL6008360 0.87 CCR5 (0.69) CCR5
SCHEMBL6006892 0.87 CCR5 (0.75) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716156-A2 CHEMOKINE CCR5 RECEPTOR MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2006-11-02 EP claimed
WO-2005075484-A2 CHEMOKINE CCR5 RECEPTOR MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-08-18 WO claimed