SCHEMBL6007316

SCHEMBL6007316

CCCCC1CN(CC2CCCCC2)C(=O)OC12CCN(C1CCN(C(=O)c3ccc(SC)cc3OC)CC1)CC2

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 18/20 0.66
LMNA P02545 1/20 0.45
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6008111 0.90 CCR5 (0.68) CCR5KCNH2
SCHEMBL6008147 0.85 CCR5 (0.74) CCR5KCNH2
SCHEMBL6008972 0.83 CCR5 (0.71) CCR5KCNH2
SCHEMBL6008609 0.82 CCR5 (0.70) CCR5KCNH2
SCHEMBL6008081 0.82 CCR5 (0.77) CCR5KCNH2
SCHEMBL6007349 0.82 CCR5 (0.81) CCR5KCNH2
SCHEMBL6005520 0.82 CCR5 (0.71) CCR5KCNH2
SCHEMBL6006159 0.81 CCR5 (0.75) CCR5KCNH2
SCHEMBL6008294 0.81 CCR5 (0.73) CCR5KCNH2
SCHEMBL6008366 0.81 CCR5 (0.84) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716156-A2 CHEMOKINE CCR5 RECEPTOR MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2006-11-02 EP claimed
WO-2005075484-A2 CHEMOKINE CCR5 RECEPTOR MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-08-18 WO claimed