SCHEMBL6007717

SCHEMBL6007717

CCCCC1CN(CC2CCCCC2)C(=O)OC12CCN(C1CCN(C(=O)c3c(-c4ccccc4Cl)noc3C)CC1)CC2

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 18/20 0.71
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
KCNH2 Q12809 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6008136 0.91 CCR5 (0.75) CCR5KCNH2
SCHEMBL6008161 0.88 CCR5 (0.85) CCR5KCNH2
SCHEMBL6008871 0.86 CCR5 (0.91) CCR5
SCHEMBL6007296 0.86 CCR5 (0.80) CCR5KCNH2
SCHEMBL6009138 0.84 CCR5 (0.80) CCR5KCNH2
SCHEMBL6008197 0.84 CCR5 (0.78) CCR5KCNH2
SCHEMBL4465187 0.83 CCR5 (1.00) CCR5
SCHEMBL4458249 0.83 CCR5 (1.00) CCR5
SCHEMBL4458255 0.83 CCR5 (1.00) CCR5
SCHEMBL6006949 0.83 CCR5 (0.98) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716156-A2 CHEMOKINE CCR5 RECEPTOR MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2006-11-02 EP claimed
WO-2005075484-A2 CHEMOKINE CCR5 RECEPTOR MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-08-18 WO claimed