SCHEMBL6008370

SCHEMBL6008370

CCCCC1N(CC2CCCCC2)C(=O)OC12CCN(C1CCN(C(=O)CCN3CCOCC3)CC1)CC2

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 15/20 0.64
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HIF1A Q16665 1/20 0.37
GAA P10253 1/20 0.37
CTSD P07339 1/20 0.35
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6006856 0.84 CCR5 (0.74) CCR5MEN1KMT2A
SCHEMBL6008248 0.83 CCR5 (0.72) CCR5
SCHEMBL6008042 0.81 CCR5 (0.74) CCR5ALDH1A1MAPTKDM4EHIF1A
SCHEMBL6009251 0.81 CCR5 (0.63) CCR5
SCHEMBL6007019 0.81 CCR5 (0.67) CCR5ALDH1A1
SCHEMBL6007098 0.80 CCR5 (0.77) CCR5
SCHEMBL6006841 0.80 CCR5 (0.65) CCR5
SCHEMBL6005547 0.79 CCR5 (0.81) CCR5KMT2AALDH1A1KDM4E
SCHEMBL6007299 0.79 CCR5 (0.76) CCR5KMT2A
SCHEMBL6009206 0.79 CCR5 (0.61) CCR5MEN1KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716156-A2 CHEMOKINE CCR5 RECEPTOR MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2006-11-02 EP claimed
WO-2005075484-A2 CHEMOKINE CCR5 RECEPTOR MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-08-18 WO claimed