SCHEMBL6011005

SCHEMBL6011005

FC(F)(F)Oc1ccc(/C=C/C2CCNCC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.45
CYP2D6 P10635 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
PIM1 P11309 1/20 0.41
PIM2 Q9P1W9 1/20 0.41
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
HTR2C P28335 1/20 0.40
MMP1 P03956 1/20 0.38
MMP3 P08254 1/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
MMP13 P45452 1/20 0.38
MMP14 P50281 1/20 0.38
NISCH Q9Y2I1 1/20 0.37
MAOB P27338 4/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27697688 0.84 EPHX1 (0.47) EPHX1CYP2D6HRH3PIM1PIM2
SCHEMBL6009169 0.80 MAOB (0.55) CYP2D6MAOBHDAC1HDAC8KDM1A
SCHEMBL9562264 0.80 MAOB (0.55) CYP2D6MAOBHDAC1HDAC8KDM1A
SCHEMBL9562365 0.80 MAOB (0.55) HRH3HTR2CMAOBHDAC1HDAC8
SCHEMBL9562361 0.80 MAOB (0.55) HRH3HTR2CMAOBHDAC1HDAC8
SCHEMBL6011007 0.78 HTR1A (0.46) KDM1A
Hydrochloric Acid SCHEMBL19994632 0.78 HTR2C (0.54) HRH3HTR2CMAOBHDAC1HDAC8
Hydrochloric Acid SCHEMBL19994635 0.78 HTR2C (0.54) HRH3HTR2CMAOBHDAC1HDAC8
SCHEMBL5213208 0.77 MAOB (0.51) MAOB
SCHEMBL9060986 0.74 HRH3 (0.38) CYP2D6HRH3PIM1PIM2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1785415-B1 PIPERIDINE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF ASTELLAS PHARMA INC (JP) 2012-05-02 EP disclosed
EP-1785415-A1 PIPERIDINE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Astellas Pharma Inc. (JP) 2007-05-16 EP disclosed