SCHEMBL6015272

SCHEMBL6015272

CCCOc1ccc(C(CC)(CC)c2ccc(CCC(C)(C)O)c(C)c2)cc1C

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
VDR P11473 13/20 0.59
HDAC3 O15379 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
AR P10275 6/20 0.47
ESR1 P03372 5/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5159678 0.87 VDR (0.54) VDRHDAC3HDAC6ARESR1
SCHEMBL5156660 0.85 HDAC6 (0.52) VDRHDAC3HDAC6ARESR1
SCHEMBL5155789 0.84 HDAC6 (0.52) VDRHDAC3HDAC6ARESR1
SCHEMBL5154482 0.83 VDR (0.77) VDRHDAC3HDAC6AR
SCHEMBL5153777 0.82 VDR (0.78) VDRAR
SCHEMBL1052998 0.82 VDR (0.78) VDRAR
SCHEMBL1057856 0.81 VDR (0.46) VDRHDAC3HDAC6ARESR1
SCHEMBL5155829 0.80 VDR (0.47) VDRHDAC3HDAC6ARESR1
SCHEMBL1053011 0.79 ESR1 (0.65) VDRARESR1
SCHEMBL5159121 0.78 ESR1 (0.49) VDRHDAC3HDAC6ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1675812-A2 BRIDGED RING STRUCTURES AS PHARMACEUTICAL AGENTS X-Ceptor Therapeutics, Inc. (US) 2006-07-05 EP disclosed
WO-2005037755-A2 BRIDGED RING STRUCTURES AS PHARMACEUTICAL AGENTS X-CEPTOR THERAPEUTICS, INC. (US) 2005-04-28 WO disclosed