SCHEMBL6015589

SCHEMBL6015589

COc1cc(C)ccc1-c1nnc(SCc2ccccn2)[nH]1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.52
CYP2E1 P05181 5/20 0.52
CYP2C8 P10632 5/20 0.52
CYP2D6 P10635 5/20 0.52
CYP2C9 P11712 5/20 0.52
CYP2B6 P20813 5/20 0.52
CYP2C19 P33261 5/20 0.52
CYP3A4 P08684 4/20 0.52
RAB9A P51151 4/20 0.49
NPC1 O15118 3/20 0.49
LMNA P02545 2/20 0.49
ALDH1A1 P00352 3/20 0.43
MAPT P10636 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
SYK P43405 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 1/20 0.41
HTT P42858 1/20 0.41
GLA P06280 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6015582 0.89 CYP1A2 (0.57) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL645267 0.88 RAB9A (0.63) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL6015602 0.87 NPC1 (0.47) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL6015595 0.87 DAO (0.38) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL6015599 0.86 CYP1A2 (0.56) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL6015605 0.83 CYP1A2 (0.57) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL6015585 0.81 NPC1 (0.53) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL1378355 0.80 NPC1 (0.78) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL6015614 0.80 PDE2A (0.39) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL6015598 0.79 CYP1A2 (0.54) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054526-A2 CHEMOSENSORY RECEPTOR LIGAND-BASED THERAPIES ELCELYX THERAPEUTICS, INC. (US) 2012-04-26 WO disclosed