SCHEMBL6015636

SCHEMBL6015636

CN(C)S(=O)(=O)c1ccc2c(C=O)c[nH]c2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.53
ALDH1A1 P00352 8/20 0.52
KDM4E B2RXH2 4/20 0.52
MAPT P10636 3/20 0.52
PLG P00747 1/20 0.47
PLAU P00749 1/20 0.47
IMPDH2 P12268 1/20 0.46
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
LMNA P02545 2/20 0.41
HTT P42858 2/20 0.41
GAA P10253 2/20 0.41
PLA2G1B P04054 1/20 0.41
HPGD P15428 1/20 0.41
ATG4B Q9Y4P1 1/20 0.41
CCNT1 O60563 1/20 0.40
CDK9 P50750 1/20 0.40
HASPIN Q8TF76 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31129989 1.00 CYP2A6 (0.53) CYP2A6ALDH1A1KDM4EMAPTPLG
SCHEMBL29956133 0.88 MAPT (0.60) CYP2A6ALDH1A1KDM4EMAPTIMPDH2
SCHEMBL14832262 0.88 MAPT (0.60) CYP2A6ALDH1A1KDM4EMAPTIMPDH2
SCHEMBL31129913 0.80 ALDH1A1 (0.46) ALDH1A1KDM4EMAPTLMNAHTT
SCHEMBL29935657 0.73 PIM3 (0.65) CYP2A6ALDH1A1KDM4EMAPTPLG
SCHEMBL1049957 0.73 PIM3 (0.65) CYP2A6ALDH1A1KDM4EMAPTPLG
SCHEMBL15902102 0.71 ALDH1A1 (0.58) CYP2A6ALDH1A1KDM4EMAPTPLG
SCHEMBL31130039 0.71 MAPT (0.54) ALDH1A1KDM4EMAPTLMNAHTT
SCHEMBL9377060 0.71 CYP2A6 (0.66) CYP2A6ALDH1A1KDM4EMAPTPLG
SCHEMBL29956305 0.71 CYP2A6 (0.66) CYP2A6ALDH1A1KDM4EMAPTPLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP disclosed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO disclosed