SCHEMBL6015941

SCHEMBL6015941

COCCC(N)c1ccc2cc[nH]c2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.47
POLB P06746 1/20 0.47
MAPK1 P28482 1/20 0.47
KMT2A Q03164 1/20 0.47
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TSHR P16473 1/20 0.40
AHR P35869 3/20 0.40
CMA1 P23946 1/20 0.40
TYR P14679 1/20 0.40
PDE2A O00408 1/20 0.38
ESR1 P03372 1/20 0.37
MAOA P21397 1/20 0.37
ENPP2 Q13822 2/20 0.37
CYP2A6 P11509 1/20 0.37
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19036434 0.79 AHR (0.43) MEN1POLBMAPK1KMT2AKDM4E
SCHEMBL3870893 0.76 MEN1 (0.47) MEN1POLBMAPK1KMT2AKDM4E
SCHEMBL12497995 0.76 MEN1 (0.47) MEN1POLBMAPK1KMT2AKDM4E
SCHEMBL16649859 0.76 MEN1 (0.47) MEN1POLBMAPK1KMT2AKDM4E
SCHEMBL11833422 0.75 MEN1 (0.55) MEN1POLBMAPK1KMT2AKDM4E
SCHEMBL27601520 0.75
SCHEMBL23342531 0.72 MEN1 (0.51) MEN1POLBMAPK1KMT2ATAS1R3
SCHEMBL83970 0.72 AHR (0.50) MEN1POLBMAPK1KMT2AKDM4E
SCHEMBL21164488 0.71 MEN1 (0.46) MEN1POLBMAPK1KMT2ATAS1R3
SCHEMBL27601642 0.71 ALDH1A1 (0.53) MEN1KMT2AKDM4EALDH1A1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed
CN-1636005-A Benzothiazinone and benzoxazinone compounds KNOLL AG (DE) 2005-07-06 CN disclosed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP disclosed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO disclosed