SCHEMBL6015958

SCHEMBL6015958

CN(C)Cc1c(OCCN2CCOCC2)ccc2[c]c[nH]c12

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
BRD4 O60885 1/20 0.41
POLB P06746 2/20 0.40
DRD1 P21728 1/20 0.38
DRD4 P21917 1/20 0.38
DRD5 P21918 1/20 0.38
MAOB P27338 1/20 0.38
SYK P43405 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
KDM4E B2RXH2 1/20 0.36
P2RY12 Q9H244 1/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016041 0.89 SMN1; SMN2 (0.43) TSHRPOLBSMN1; SMN2KDM4E
SCHEMBL6016076 0.89 SMN1; SMN2 (0.43) TSHRPOLBSMN1; SMN2KDM4E
SCHEMBL6015789 0.78
SCHEMBL6015751 0.77
SCHEMBL6015772 0.75 HPGD (0.51) TSHRSMN1; SMN2ALDH1A1MAPTHTT
SCHEMBL6015642 0.73
SCHEMBL7624616 0.73 PIM1 (0.35)
SCHEMBL6015721 0.72
SCHEMBL6016018 0.69 KDM4E (0.55) TSHRALDH1A1KDM4ENPC1
SCHEMBL6015938 0.69 TSHR (0.51) TSHRPOLBDRD1DRD4DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US claimed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP claimed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP disclosed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO disclosed