SCHEMBL6016366

SCHEMBL6016366

Cc1ccc(-c2nc(OCCN3CCOCC3)ncc2N(C)C(=O)C(C)(C)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.51
TACR3 P29371 8/20 0.43
CYP3A4 P08684 5/20 0.41
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HIF1A Q16665 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016365 0.88 TACR1 (0.63) TACR1TACR3CYP3A4
SCHEMBL6882076 0.84 TACR1 (0.55) TACR1TACR3CYP3A4
SCHEMBL6871218 0.83 TACR1 (0.46) TACR1TACR3CYP3A4
SCHEMBL5802838 0.82 TACR1 (0.49) TACR1TACR3
SCHEMBL6664695 0.81 TACR1 (0.47) TACR1TACR3CYP3A4
SCHEMBL6876208 0.81 TACR1 (0.44) TACR1TACR3CYP3A4
SCHEMBL6881887 0.80 TACR1 (0.47) TACR1TACR3
SCHEMBL6664699 0.79 TACR1 (0.57) TACR1TACR3CYP3A4
SCHEMBL7760176 0.76 TACR1 (0.78) TACR1TACR3CYP3A4
SCHEMBL6019565 0.73 TACR1 (0.49) TACR1TACR3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187815-B1 4-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-02-08 EP disclosed