SCHEMBL6664699

SCHEMBL6664699

Cc1ccc(-c2cc(N(C)CCN3CCOCC3)ncc2N(C)C(=O)C(C)(C)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 20/20 0.57
TACR3 P29371 12/20 0.55
CYP3A4 P08684 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4134901 0.88 TACR1 (0.71) TACR1TACR3CYP3A4
SCHEMBL23385302 0.87 TACR1 (0.60) TACR1TACR3CYP3A4
SCHEMBL6664695 0.85 TACR1 (0.47) TACR1TACR3CYP3A4
SCHEMBL7760176 0.84 TACR1 (0.78) TACR1TACR3CYP3A4
SCHEMBL6016366 0.79 TACR1 (0.51) TACR1TACR3CYP3A4
SCHEMBL6521393 0.79 TACR1 (0.55) TACR1TACR3CYP3A4
SCHEMBL23385207 0.79 TACR1 (0.58) TACR1TACR3CYP3A4
SCHEMBL1870486 0.78 TACR1 (0.72) TACR1TACR3CYP3A4
SCHEMBL6019571 0.78 TACR1 (0.62) TACR1TACR3CYP3A4
SCHEMBL15227973 0.76 TACR1 (0.55) TACR1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1035115-B1 4-Phenylpyridine derivatives and their use as NK-1 receptor antagonists HOFFMANN LA ROCHE (CH) 2004-09-29 EP claimed