SCHEMBL6016939

SCHEMBL6016939

N#Cc1ccccc1Cn1c(F)nc2ccc(F)cc2c1=O

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 0.63
DPP4 P27487 9/20 0.63
NOX4 Q9NPH5 1/20 0.49
MAPK14 Q16539 1/20 0.46
GRIN1 Q05586 3/20 0.45
GRIN2B Q13224 3/20 0.45
KMT2A Q03164 1/20 0.43
MAPT P10636 1/20 0.43
CASR P41180 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3425489 0.89 CYP3A4 (0.61) CYP3A4DPP4NOX4MAPK14GRIN1
SCHEMBL3425219 0.78 DPP4 (1.00) CYP3A4DPP4
SCHEMBL3421937 0.78 DPP4 (1.00) CYP3A4DPP4
SCHEMBL3425757 0.77 CYP3A4 (0.63) CYP3A4DPP4NOX4GRIN1GRIN2B
SCHEMBL3428161 0.75 DPP4 (0.61) CYP3A4DPP4NOX4GRIN1GRIN2B
SCHEMBL6216570 0.73
SCHEMBL3423901 0.73 DPP4 (0.57) CYP3A4DPP4NOX4KMT2AMAPT
SCHEMBL3425852 0.73 CYP3A4 (0.63) CYP3A4DPP4NOX4GRIN1GRIN2B
SCHEMBL3426403 0.70 NOX4 (0.47) CYP3A4DPP4NOX4GRIN1GRIN2B
SCHEMBL3423226 0.70 DPP4 (0.64) CYP3A4DPP4NOX4MAPK14GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1608317-A4 DIPEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2006-12-27 EP claimed
EP-1608317-A2 DIPEPTIDYL PEPTIDASE INHIBITORS Takeda San Diego, Inc. (US) 2005-12-28 EP claimed
WO-2004087053-A2 DIPEPTIDYL PEPTIDASE INHIBITORS SYRRX, INC. (US) 2004-10-14 WO claimed