SCHEMBL6017748

SCHEMBL6017748

Nc1nc(-c2ccccc2)nc2cccc(OC(F)c3ccccc3)c12

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHFR P00374 5/20 0.46
DCPS Q96C86 4/20 0.41
CYP1A1 P04798 5/20 0.40
CYP1A2 P05177 5/20 0.40
CYP1B1 Q16678 5/20 0.40
KCNH2 Q12809 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2125491 0.78 ABCG2 (0.51) DHFRDCPSCYP1A1CYP1A2CYP1B1
SCHEMBL1154543 0.73 DHFR (0.75) DHFRDCPSKCNH2
SCHEMBL1155243 0.73 DHFR (0.75) DHFRDCPSKCNH2
SCHEMBL1154243 0.73 DHFR (0.75) DHFRDCPSKCNH2
SCHEMBL1154437 0.72 DHFR (0.60) DHFRDCPSKCNH2
SCHEMBL20483820 0.68 ELANE (0.49) DHFRCYP1A1CYP1A2CYP1B1
SCHEMBL29593101 0.66 CYP1A1 (0.77) DCPSCYP1A1CYP1A2CYP1B1
SCHEMBL1395347 0.66 CYP1A1 (0.77) DCPSCYP1A1CYP1A2CYP1B1
SCHEMBL1154842 0.66 DHFR (0.70) DHFRDCPSKCNH2
SCHEMBL1154943 0.66 DHFR (0.74) DHFRDCPSKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664028-A1 QUINAZOLINE DERIVATIVES AS TYROSINE KINASE INHIBITORS AstraZeneca AB (SE) 2006-06-07 EP disclosed
WO-2005026151-A1 QUINAZOLINE DERIVATIVES AS TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2005-03-24 WO disclosed