SCHEMBL6019264

SCHEMBL6019264

NC(=O)c1ccc2[nH]ncc2c1.O=C(N[C@@H](CCCNCc1ccccn1)C(=O)O)c1ccc(CNCc2ccccn2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 2/20 0.47
CTNNB1 P35222 2/20 0.40
WNT3A P56704 2/20 0.40
DHFR P00374 3/20 0.38
ROCK2 O75116 2/20 0.38
ROCK1 Q13464 2/20 0.38
JAK3 P52333 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
TYMS P04818 2/20 0.37
GART P22102 1/20 0.37
ATIC P31939 1/20 0.37
PADI4 Q9UM07 1/20 0.37
PADI2 Q9Y2J8 1/20 0.37
MAOB P27338 1/20 0.37
NPC1 O15118 1/20 0.36
JAK2 O60674 1/20 0.36
RAB9A P51151 1/20 0.36
FOLH1 Q04609 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27597838 1.00 CXCR4 (0.47) CXCR4CTNNB1WNT3ADHFRROCK2
SCHEMBL6018116 0.84 CXCR4 (0.53) CXCR4NPC1RAB9AFOLH1KMT2A
SCHEMBL27566287 0.84 CXCR4 (0.53) CXCR4NPC1RAB9AFOLH1KMT2A
SCHEMBL6018220 0.83 CXCR4 (0.51) CXCR4DHFRTYMSNPC1RAB9A
SCHEMBL6671573 0.82 CXCR4 (0.51) CXCR4DHFRNPC1RAB9AFOLH1
Phenylhydrazine SCHEMBL6690774 0.80 CXCR4 (0.50) CXCR4DHFRTYMSNPC1RAB9A
SCHEMBL6018262 0.77 CXCR4 (0.57) CXCR4DHFRTYMSNPC1RAB9A
SCHEMBL6840697 0.77 CXCR4 (0.46) CXCR4FOLH1KMT2AMAPK14
SCHEMBL6670076 0.76 CXCR4 (0.48) CXCR4DHFRTYMSNPC1RAB9A
Tryptamine SCHEMBL6670107 0.76 CXCR4 (0.47) CXCR4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7098215-B2 Nitrogenous compounds and antiviral drugs containing the same KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 2006-08-29 US disclosed
US-20040157818-A1 Cxcr4-antagonistic drugs composed of nitrogen-containing compound KUREHA CORPORATION (JP) 2004-08-12 US disclosed
US-20040092556-A1 Nitrogenous compounds and antiviral drugs containing the same KUREHA CORPORATION (JP) 2004-05-13 US disclosed
EP-1389460-A1 CXCR4-ANTAGONISTIC DRUGS COMPRISING NITROGEN-CONTAINING COMPOUND Kureha Chemical Industry Co., Ltd. (JP) 2004-02-18 EP disclosed
EP-1273571-A1 NITROGENOUS COMPOUNDS AND ANTIVIRAL DRUGS CONTAINING THE SAME Kureha Chemical Industry Co., Ltd. (JP) 2003-01-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040092556-A1 Nitrogenous compounds and antiviral drugs containing the same NSUN2, ZC3HAV1L, PNP CXCR4 2185/4885CTNNB1 1208/4885WNT3A 2895/4885
US-20040157818-A1 Cxcr4-antagonistic drugs composed of nitrogen-containing compound CXCR4, CXCR1, CXCR2 CXCR4 1/4885CTNNB1 352/4885WNT3A 574/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.