SCHEMBL6019933

SCHEMBL6019933

CN(CCC1CCC(CCCN2CCCCC2)CC1)C(=O)Oc1ccc(C(F)(F)F)cc1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LSS P48449 4/20 0.52
HRH3 Q9Y5N1 7/20 0.45
SLC6A4 P31645 1/20 0.45
MCHR1 Q99705 1/20 0.45
SLC6A5 Q9Y345 3/20 0.44
NAAA Q02083 1/20 0.44
LTA4H P09960 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6019936 1.00 LSS (0.52) LSSHRH3SLC6A4MCHR1SLC6A5
SCHEMBL6019946 0.92 LSS (0.55) LSSMCHR1SLC6A5NAAA
SCHEMBL6019950 0.92 LSS (0.55) LSSMCHR1SLC6A5NAAA
SCHEMBL6019452 0.90 LSS (0.51) LSSMCHR1SLC6A5NAAA
SCHEMBL6019454 0.90 LSS (0.51) LSSMCHR1SLC6A5NAAA
SCHEMBL6019222 0.90 LSS (0.49) LSSHRH3NAAA
SCHEMBL6019229 0.90 LSS (0.49) LSSHRH3NAAA
SCHEMBL4802021 0.88 LSS (0.62) LSSHRH3SLC6A4MCHR1SLC6A5
SCHEMBL4802026 0.88 LSS (0.62) LSSHRH3SLC6A4MCHR1SLC6A5
SCHEMBL6018967 0.84 LSS (0.58) LSSMCHR1SLC6A5NAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1456171-B1 SUBSTITUTED CYCLOHEXANE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-12-20 EP disclosed
US-20050272774-A1 Substituted cyclohexane derivatives ACKERMANN JEAN 2005-12-08 US disclosed
US-6953806-B2 Substituted cyclohexane derivatives HOFFMANN-LA ROCHE INC. (US) 2005-10-11 US disclosed
EP-1456171-A1 SUBSTITUTED CYCLOHEXANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2004-09-15 EP disclosed
US-20030199550-A1 Substituted cyclohexane derivatives F.HOFFMANN-LA ROCHE AG (CH) 2003-10-23 US disclosed
WO-2003053919-A1 SUBSTITUTED CYCLOHEXANE DERIVATIVES F. HOFFMANN-LA-ROCHE AG (CH) 2003-07-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050272774-A1 Substituted cyclohexane derivatives LSS, CYP51A1, CYP8B1 LSS 1/4885HRH3 3277/4885SLC6A4 4588/4885
US-20030199550-A1 Substituted cyclohexane derivatives CYP51A1, LSS, CYP46A1 LSS 2/4885HRH3 4086/4885SLC6A4 4715/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.