SCHEMBL6022247

SCHEMBL6022247

Cc1cc(CN2CCOCC2)nc(SCc2ccc(S(C)(=O)=O)cc2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
HTT P42858 3/20 0.44
NPSR1 Q6W5P4 3/20 0.44
LMNA P02545 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
JAK2 O60674 4/20 0.41
JAK3 P52333 4/20 0.41
PTK2 Q05397 4/20 0.41
HSD17B10 Q99714 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
SLC2A1 P11166 1/20 0.39
POLB P06746 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5047300 0.87 ALDH1A1 (0.48) ALDH1A1HTTNPSR1LMNAL3MBTL1
SCHEMBL5049040 0.83 ALDH1A1 (0.63) ALDH1A1HTTNPSR1LMNAL3MBTL1
SCHEMBL5045760 0.83 ALDH1A1 (0.45) ALDH1A1HTTNPSR1LMNAL3MBTL1
SCHEMBL5042312 0.77 HSD17B10 (0.46) ALDH1A1HTTNPSR1LMNAKDM4E
SCHEMBL5776873 0.74 HRH3 (0.61) ALDH1A1LMNAMAPTJAK2JAK3
SCHEMBL5042347 0.73 HSD17B10 (0.48) ALDH1A1HTTNPSR1HSD17B10CYP1A2
SCHEMBL5045968 0.72 POLB (0.46) ALDH1A1HTTKDM4EHSD17B10CYP1A2
SCHEMBL5049081 0.72 HSD17B10 (0.47) ALDH1A1HTTGAAHSD17B10CYP1A2
SCHEMBL5042209 0.71 HSD17B10 (0.46) ALDH1A1HTTGAAHSD17B10CYP1A2
SCHEMBL5050422 0.69 HTT (0.41) ALDH1A1HTTLMNAHSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1725239-A1 4-(SULFANYL-PYRIMIDIN-4-YLMETHYL)-MORPHOLINE DERIVATIVES AND RELATED COMPOUNDS AS GABA RECEPTOR LIGANDS FOR THE TREATMENT OF ANXIETY, DEPRESSION AND EPILEPSY F.HOFFMANN-LA ROCHE AG (CH) 2006-11-29 EP disclosed
WO-2005094828-A1 4- (SULFANYL-PYRIMIDIN-4-YLMETHYL) -MORPHOLINE DERIVATIVES AND RELATED COMPOUNDS AS GABA RECEPTOR LIGANDS FOR THE TREATMENT OF ANXIETY, DEPRESSION AND EPILEPSY F. HOFFMANN-LA ROCHE AG (CH) 2005-10-13 WO disclosed