SCHEMBL6025527

SCHEMBL6025527

COc1cccnc1-c1ccc(Nc2ccc3c(n2)CC(C)(C)CC3=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 3/20 0.45
MAOA P21397 2/20 0.43
MAOB P27338 2/20 0.43
GRM5 P41594 3/20 0.43
ALDH1A1 P00352 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP2C19 P33261 2/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA4 P22748 1/20 0.40
CA9 Q16790 1/20 0.40
USP2 O75604 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
GSK3B P49841 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4432470 0.80 CYP2C19 (0.51) MAP4K1MAOAMAOBGRM5ALDH1A1
SCHEMBL4427130 0.80 MAP4K1 (0.47) MAP4K1MAOAMAOBGRM5ALDH1A1
SCHEMBL4424635 0.79 MAP4K1 (0.48) MAP4K1MAOAMAOBGRM5ALDH1A1
SCHEMBL4423359 0.77 MAP4K1 (0.52) MAP4K1MAOAMAOBGRM5ALDH1A1
SCHEMBL4430358 0.76 KMT2A (0.53) MAP4K1MAOAMAOBALDH1A1NPC1
SCHEMBL4432318 0.76 CYP2C19 (0.55) MAP4K1MAOAMAOBGRM5ALDH1A1
SCHEMBL4424753 0.74 MAOA (0.55) MAP4K1MAOAMAOBGRM5ALDH1A1
SCHEMBL4430352 0.74 CYP2C19 (0.52) MAP4K1MAOAMAOBGRM5ALDH1A1
SCHEMBL4425787 0.72 MAP4K1 (0.45) MAP4K1MAOAMAOBGRM5ALDH1A1
SCHEMBL4424035 0.71 MAOA (0.44) MAP4K1MAOAMAOBGRM5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1723116-A2 TETRAHYDROQUINOLINONES AND THEIR USE AS ANTAGONISTS OF METABOTROPIC GLUTAMATE RECEPTORS Merz Pharma GmbH & Co. KGaA (DE) 2006-11-22 EP disclosed
WO-2005082856-A2 TETRAHYDROQUINOLINONES AND THEIR USE AS ANTAGONISTS OF METABOTROPIC GLUTAMATE RECEPTORS MERZ PHARMA GMBH & CO. KGAA (DE) 2005-09-09 WO disclosed